European Journal of Medicinal Chemistry
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Publication date: 5 December 2023Source: European Journal of Medicinal Chemistry, Volume 261Author(s):
European Journal of Medicinal Chemistry
Contents continued
Publication date: 5 December 2023Source: European Journal of Medicinal Chemistry, Volume 261Author(s):
European Journal of Medicinal Chemistry
Design and synthesis of pyrazole derivatives against neutrophilic inflammation
Publication date: 15 December 2023Source: European Journal of Medicinal Chemistry, Volume 262Author(s): Ko-Hua Yu, Kai-wen Tien, Wei-Chun Wang, Ching-Ho Chi, Keng-Chang Tsai, Chen-Hsi Chou, Tsong-Long Hwang, Hsin-Yi Hung
European Journal of Medicinal Chemistry
Lipidation and PEGylation strategies to prolong the <em>in vivo</em> half-life of a nanomolar EphA4 receptor antagonist
Publication date: 15 December 2023Source: European Journal of Medicinal Chemistry, Volume 262Author(s): Maricel Gomez-Soler, Erika J. Olson, Elena Rubio de la Torre, Chunxia Zhao, Ilaria Lamberto, Dillon T. Flood, Waleed Danho, Bernhard C. Lechtenberg,…
European Journal of Medicinal Chemistry
Synthetic approaches and application of clinically approved small-molecule drugs to treat hepatitis
Publication date: 15 December 2023Source: European Journal of Medicinal Chemistry, Volume 262Author(s): Zhen-Xi Niu, Peng Nie, Piet Herdewijn, Ya-Tao Wang
European Journal of Medicinal Chemistry
Design and synthesis of certain 7-Aryl-2-Methyl-3-Substituted Pyrazolo{1,5-a}Pyrimidines as multikinase inhibitors
Publication date: 15 December 2023Source: European Journal of Medicinal Chemistry, Volume 262Author(s): Mustafa A. Al-Qadhi, Heba Abdelrasheed Allam, Samar H. Fahim, Tawfeek A.A. Yahya, Fatma A.F. Ragab
European Journal of Medicinal Chemistry
Structure-based identification of new orally bioavailable BRD9-PROTACs for treating acute myelocytic leukemia
Publication date: Available online 17 October 2023Source: European Journal of Medicinal ChemistryAuthor(s): Jingyu Zhang, Haiting Duan, Renzhao Gui, Mingfei Wu, Liteng Shen, Yuheng Jin, Ao Pang, Xiaoli Yu, Shenxin Zeng, Bo Zhang, Nengming Lin, Wenhai H…
European Journal of Medicinal Chemistry
Covalent and noncovalent strategies for targeting Lys102 in HIV-1 reverse transcriptase
Publication date: 15 December 2023Source: European Journal of Medicinal Chemistry, Volume 262Author(s): Giavana R. Prucha, Sean Henry, Klarissa Hollander, Zachary J. Carter, Krasimir A. Spasov, William L. Jorgensen, Karen S. Anderson
European Journal of Medicinal Chemistry
Next generation fibroblast activation protein (FAP) targeting PET tracers – The tetrazine ligation allows an easy and convenient way to <sup>18</sup>F-labeled (4-quinolinoyl)glycyl-2-cyanopyrrolidines
Publication date: 15 December 2023Source: European Journal of Medicinal Chemistry, Volume 262Author(s): Christian B.M. Poulie, Vladimir Shalgunov, Filipe Elvas, Yentl Van Rymenant, Euy-Sung Moon, Umberto Maria Battisti, Joni De Loose, Ingrid De Meester…
European Journal of Medicinal Chemistry
Design, synthesis and biological evaluation of novel dihydroquinolin-4(1<em>H</em>)-one derivatives as novel tubulin polymerization inhibitors
Publication date: 15 December 2023Source: European Journal of Medicinal Chemistry, Volume 262Author(s): Yuchen Tan, Han Hu, Wenjian Zhu, Tao Wang, Tian Gao, Hongqi Wang, Jian Chen, Jinyi Xu, Shengtao Xu, Huajian Zhu