Bioorganic & Medicinal Chemistry
Graphical Abstract Contents Continued
Publication date: 1 November 2022Source: Bioorganic & Medicinal Chemistry, Volume 73Author(s):
Bioorganic & Medicinal Chemistry
Guanidine-based β amyloid precursor protein cleavage enzyme 1 (BACE-1) inhibitors for the Alzheimer’s disease (AD): A review
Publication date: 15 November 2022Source: Bioorganic & Medicinal Chemistry, Volume 74Author(s): Pinky Gehlot, Sunil Kumar, Vivek Kumar Vyas, Bhanwar Singh Choudhary, Manish Sharma, Ruchi Malik
Bioorganic & Medicinal Chemistry
Graphical abstract TOC
Publication date: 1 November 2022Source: Bioorganic & Medicinal Chemistry, Volume 73Author(s):
Bioorganic & Medicinal Chemistry
Discovery of a new class of valosine containing protein (VCP/P97) inhibitors for the treatment of colorectal cancer
Publication date: 15 November 2022Source: Bioorganic & Medicinal Chemistry, Volume 74Author(s): Xueyuan Wang, Tiantian Wen, Hang Miao, Wenjiao Hu, Meng Lei, Yongqiang Zhu
Bioorganic & Medicinal Chemistry
Discovery of selective covalent cathepsin K inhibitors containing novel 4-cyanopyrimidine warhead based on quantum chemical calculations and binding mode analysis
Publication date: 15 November 2022Source: Bioorganic & Medicinal Chemistry, Volume 74Author(s): Yihe Jia, Ke Wang, Huifang Wang, Botao Zhang, Kan Yang, Zhilan Zhang, Haijuan Dong, Jinxin Wang
Bioorganic & Medicinal Chemistry
Design, synthesis and biological evaluation of novel 4-aminopiperidine derivatives as SMO/ERK dual inhibitors
Publication date: 15 November 2022Source: Bioorganic & Medicinal Chemistry, Volume 74Author(s): Jing-Jing Zhang, Wanwan Zhang, Lei Zhang, Mengxuan Hu, Qi-Jie Xu, Yungen Xu
Bioorganic & Medicinal Chemistry
Design, synthesis and antitumor efficacy evaluation of a series of novel β-elemene-based macrocycles
Publication date: 15 November 2022Source: Bioorganic & Medicinal Chemistry, Volume 74Author(s): Xiang Qi, Songwei Jiang, Zi Hui, Yuan Gao, Yang Ye, Frédéric Lirussi, Carmen Garrido, Li Xu, Xingrui He, Renren Bai, Xiang-Yang Ye, Tian Xie
Bioorganic & Medicinal Chemistry
Design, synthesis and biological evaluation of novel pyrazinone derivatives as PI3K/HDAC dual inhibitors
Publication date: 15 November 2022Source: Bioorganic & Medicinal Chemistry, Volume 74Author(s): Zi-Xiao Wang, Shuai Wang, Xue-Peng Qiao, Wen-Bo Li, Jian-Tao Shi, Yi-Ru Wang, Shi-Wu Chen
Bioorganic & Medicinal Chemistry
<em>meta</em>-Ureidophenoxy-1,2,3-triazole hybrid as a novel scaffold for promising HepG2 hepatocellular carcinoma inhibitors: Synthesis, biological evaluation and molecular docking studies
Publication date: 15 November 2022Source: Bioorganic & Medicinal Chemistry, Volume 74Author(s): Panupun Limpachayaporn, Sopon Nuchpun, Jitnapa Sirirak, Purin Charoensuksai, Pawaris Wongprayoon, Natthaya Chuaypen, Pisit Tangkijvanich, Apichart Suksamrarn
Bioorganic & Medicinal Chemistry
Development of carbohydrate based next-generation anti-pertussis vaccines
Publication date: Available online 17 October 2022Source: Bioorganic & Medicinal ChemistryAuthor(s): Peng Wang, Sherif Ramadan, Purnima Dubey, Rajendar Deora, Xuefei Huang