Bioorganic & Medicinal Chemistry

Synthesis and Biological Evaluation of <em>tert</em>-Butyl Ester and Ethyl Ester Prodrugs of <em>L</em>-γ-Methyleneglutamic Acid Amides for Cancer

Publication date: Available online 21 December 2022Source: Bioorganic & Medicinal ChemistryAuthor(s): Md Imdadul H. Khan, Fakhri Mahdi, Patrice Penfornis, Nicholas S. Akins, Md Imran Hossain, Seong Jong Kim, Suresh P. Sulochana, Amna T. Adam, Tristan D…

By ScienceDirect Publication: Bioorganic & Medicinal Chemistry, ago

Bivalent dopamine agonists with co-operative binding and functional activities at dopamine D2 receptors, modulate aggregation and toxicity of alpha synuclein protein

Publication date: Available online 16 December 2022Source: Bioorganic & Medicinal ChemistryAuthor(s): Bidyut Dinda, Banibrata Das, Swati Biswas, Horrick Sharma, Christopher Armstrong, Deepthi Yedlapudi, Tamara Antonio, Maarten Reith, Aloke K. Dutta

By ScienceDirect Publication: Bioorganic & Medicinal Chemistry, ago

Corrigendum to “A novel survivin dimerization inhibitor without a labile hydrazone linker induces spontaneous apoptosis and synergizes with docetaxel in prostate cancer cells” [Bioorg. Med. Chem. 65 (2022) 116761]

Publication date: Available online 12 December 2022Source: Bioorganic & Medicinal ChemistryAuthor(s): Robert Peery, Qingbin Cui, Kwaku Kyei-Baffour, Sophia Josephraj, Caoqinglong Huang, Zizheng Dong, Mingji Dai, Jian-Ting Zhang, Jing-Yuan Liu

By ScienceDirect Publication: Bioorganic & Medicinal Chemistry, ago