Bioorganic & Medicinal Chemistry
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Publication date: 15 February 2023Source: Bioorganic & Medicinal Chemistry, Volume 80Author(s):
Bioorganic & Medicinal Chemistry
Design, synthesis and biological evaluation of KRAS<sup>G12C</sup>-PROTACs
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry, Volume 78Author(s): Xiaoyi Zhang, Tong Zhao, Minghao Sun, Pei Li, Mengzhen Lai, Lingfeng Xie, Jiaying Chen, Jian Ding, Hua Xie, Jinpei Zhou, Huibin Zhang
Bioorganic & Medicinal Chemistry
The effect of diphenylethane side-chain substituents on dibenzocyclohexadiene formation and their inhibition of α-synuclein aggregation <em>in vitro</em>
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry, Volume 78Author(s): Gabriel Bernardes, Omer Munir, Ed S. Krol
Bioorganic & Medicinal Chemistry
Design, synthesis, and biological evaluation of quinoxalinone derivatives as potent BRD4 inhibitors
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry, Volume 78Author(s): Kai-Yan Xu, Xue-Ting Wang, Lei Cheng, Qi-Hang Cui, Jian-Tao Shi, Li-Wen Zhang, Shi-Wu Chen
Bioorganic & Medicinal Chemistry
Synthesis and biophysical properties of tetravalent PEG-conjugated antisense oligonucleotide
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry, Volume 78Author(s): Taslima Rahman Chowdhury, Tahia Taufiq, Kenta Ishida, Md Ariful Islam, Yuuya Kasahara, Takashi Osawa, Satoshi Obika
Bioorganic & Medicinal Chemistry
Auranofin inhibits virulence pathways in <em>Pseudomonas aeruginosa</em>
Publication date: Available online 12 January 2023Source: Bioorganic & Medicinal ChemistryAuthor(s): Joey Kuok Hoong Yam, Leon Zhen Wei Tan, Ziyan Hong, May Margarette Santillan Salido, Bau Yi Woo, Adeline Mei Hui Yong, Casandra Ai Zhu Tan, Sam Fong Ya…
Bioorganic & Medicinal Chemistry
Discovery of aromatic 2-(3-(methylcarbamoyl) guanidino)-N-aylacetamides as highly potent chitinase inhibitors
Publication date: Available online 12 January 2023Source: Bioorganic & Medicinal ChemistryAuthor(s): Zhixiang Zhao, Fang Li, Wei Chen, Qing Yang, Huizhe Lu, Jianjun Zhang
Bioorganic & Medicinal Chemistry
Synthesis and Discovery of Baylis-Hillman Adducts as Potent and Selective Thioredoxin Reductase Inhibitors for Cancer Treatment
Publication date: Available online 12 January 2023Source: Bioorganic & Medicinal ChemistryAuthor(s): Yi-Lin He, Miao Zhong, Zi-Long Song, Yu-Kai Shen, Lanning Zhao, Jianguo Fang
Bioorganic & Medicinal Chemistry
Design, synthesis and biological evaluation of novel 9-<em>N</em>-substituted-13-alkylberberine derivatives from Chinese medicine as anti-hepatocellular carcinoma agents
Publication date: Available online 8 January 2023Source: Bioorganic & Medicinal ChemistryAuthor(s): Jichao Chen, Yiping Duan, Kan Yang, Jiahe Wang, Junjie Yan, Chenglei Gu, Shanglong Wang, Zheying Zhu, E-Hu Liu, Jinyi Xu
Bioorganic & Medicinal Chemistry
2-Anilino-4-(1-methyl-1<em>H</em>-pyrazol-4-yl)pyrimidine-derived CDK2 Inhibitors as Anticancer Agents: Design, Synthesis & Evaluation
Publication date: Available online 11 January 2023Source: Bioorganic & Medicinal ChemistryAuthor(s): Biruk Sintayehu Fanta, Laychiluh Mekonnen, Sunita K.C. Basnet, Theodosia Teo, Jimma Lenjisa, Nishat Z. Khair, Lianmeng Kou, Solomon Tadesse, Matthew J….