Bioorganic & Medicinal Chemistry
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Publication date: 15 March 2023Source: Bioorganic & Medicinal Chemistry, Volume 82Author(s):
Bioorganic & Medicinal Chemistry
Graphical abstract TOC
Publication date: 15 March 2023Source: Bioorganic & Medicinal Chemistry, Volume 82Author(s):
Bioorganic & Medicinal Chemistry
Design, synthesis and biological evaluation of the tumor hypoxia-activated PROTACs bearing caged CRBN E3 ligase ligands
Publication date: 15 March 2023Source: Bioorganic & Medicinal Chemistry, Volume 82Author(s): Weiyan Cheng, Shasha Li, Siyuan Han, Ruoyang Miao, Suhua Wang, Chunxia Liu, Han Wei, Xin Tian, Xiaojian Zhang
Bioorganic & Medicinal Chemistry
Synthesis, biological activity and mechanism of action of novel allosecurinine derivatives as potential antitumor agents
Publication date: 15 March 2023Source: Bioorganic & Medicinal Chemistry, Volume 82Author(s): Xin-Liang Xu, Jin-Xia Lan, Hao Huang, Wei Dai, Xiao-Peng Peng, Sheng-Lan Liu, Wei-Ming Chen, Le-Jun Huang, Jun Liu, Xiao-Jun Li, Jun-Lin Zeng, Xian-Hua Huang, …
Bioorganic & Medicinal Chemistry
A novel selective estrogen receptor degrader induces cell cycle arrest in breast cancer via ERα degradation and the autophagy-lysosome pathway
Publication date: 15 March 2023Source: Bioorganic & Medicinal Chemistry, Volume 82Author(s): Jiawei Zhou, Rong Shen, Jing Liu, Xiangping Deng, Lilan Xin, Hai-Bing Zhou, Jian Huang
Bioorganic & Medicinal Chemistry
Novel xanthone antibacterials: Semi-synthesis, biological evaluation, and the action mechanisms
Publication date: Available online 8 March 2023Source: Bioorganic & Medicinal ChemistryAuthor(s): Lu Yan, Ting Guan, Shaobing Wang, Cui Zhou, Meizhu Wang, Xiaoyang Wang, Keyu Zhang, Xiangan Han, Jinchao Lin, Qun Tang, Chunmei Wang, Wen Zhou
Bioorganic & Medicinal Chemistry
<sup>18</sup>F-Labeled <em>o</em>‑aminopyridyl alkynyl radioligands targeting colony-stimulating factor 1 receptor for neuroinflammation imaging
Publication date: Available online 8 March 2023Source: Bioorganic & Medicinal ChemistryAuthor(s): Xiaodan An, Jingqi Wang, Linjiang Tong, Xiaojun Zhang, Hualong Fu, Jinming Zhang, Hua Xie, Yiyun Huang, Hongmei Jia
Bioorganic & Medicinal Chemistry
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Publication date: 1 March 2023Source: Bioorganic & Medicinal Chemistry, Volume 81Author(s):
Bioorganic & Medicinal Chemistry
There’s more to enzyme antagonism than inhibition
Publication date: Available online 5 March 2023Source: Bioorganic & Medicinal ChemistryAuthor(s): Brian P. Callahan, Zihan Xu
Bioorganic & Medicinal Chemistry
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Publication date: 1 March 2023Source: Bioorganic & Medicinal Chemistry, Volume 81Author(s):