Bioorganic & Medicinal Chemistry Letters
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Publication date: 15 October 2022Source: Bioorganic & Medicinal Chemistry Letters, Volume 74Author(s):
Bioorganic & Medicinal Chemistry Letters
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Publication date: 15 October 2022Source: Bioorganic & Medicinal Chemistry Letters, Volume 74Author(s):
Bioorganic & Medicinal Chemistry Letters
Discovery of 3,4-dihydropyrimido[4,5-<em>d</em>]pyrimidin-2(1<em>H</em>)-one and 3,4-dihydropyrido[2,3-<em>d</em>]pyrimidin-2(1<em>H</em>)-one derivatives as novel ENPP1 inhibitors
Publication date: 1 November 2022Source: Bioorganic & Medicinal Chemistry Letters, Volume 75Author(s): Jae Eun Jung, Yunseong Jang, Hee Jin Jeong, Sung Joon Kim, Kichul Park, Do Hee Oh, Ahran Yu, Chan Sun Park, Seo-Jung Han
Bioorganic & Medicinal Chemistry Letters
Nitro compounds against trypanosomatidae parasites: Heroes or villains?
Publication date: 1 November 2022Source: Bioorganic & Medicinal Chemistry Letters, Volume 75Author(s): Paulo Fernando da Silva Santos-Júnior, Leandro Rocha Silva, Lucindo José Quintans-Júnior, Edeildo Ferreira da Silva-Júnior
Bioorganic & Medicinal Chemistry Letters
Ultrasensitive, rapid, and highly specific detection of microRNAs based on PER-CRISPR/CAS
Publication date: 15 October 2022Source: Bioorganic & Medicinal Chemistry Letters, Volume 74Author(s): Ze Wang, Hongguo Wei, Shengjun Bu, Xue Li, Hongyu Zhou, Wenhui Zhang, Jiayu Wan
Bioorganic & Medicinal Chemistry Letters
Targeting non-alcoholic fatty liver disease: Design, X-ray co-crystal structure and synthesis of ‘first-in-kind’ inhibitors of serine/threonine kinase25
Publication date: 1 November 2022Source: Bioorganic & Medicinal Chemistry Letters, Volume 75Author(s): Scarlett Kiyeleko, Sofiane Hocine, Giséle Mautino, Mélaine Kuenemann, Agata Nawrotek, Linda Miallau, Laurent-Michel Vuillard, Olivier Mirguet, Andras…
Bioorganic & Medicinal Chemistry Letters
Identification of the gossypol derivatives as androgen receptor inhibitor
Publication date: 1 November 2022Source: Bioorganic & Medicinal Chemistry Letters, Volume 75Author(s): Rongyu Zhang, Meng Wu, Tongxiang Cao, Kui Luo, Fangjiao Huang, Ruoying Zhang, Zhipeng Huang, Jinming Zhou, Yongdong Wang, Shifa Zhu
Bioorganic & Medicinal Chemistry Letters
Aiming to improve binding of porphyrin diphenyl guanidinium conjugates to guanine-quadruplexes: When size matters
Publication date: 1 November 2022Source: Bioorganic & Medicinal Chemistry Letters, Volume 75Author(s): Nikolina Stipaničev, Konstantin Raabe, Isabel Rozas
Bioorganic & Medicinal Chemistry Letters
The discovery of BMS-737 as a potent, CYP17 lyase-selective inhibitor for the treatment of castration-resistant prostate cancer
Publication date: 1 November 2022Source: Bioorganic & Medicinal Chemistry Letters, Volume 75Author(s): Chetan Padmakar Darne, Upender Velaparthi, Mark Saulnier, David Frennesson, Peiying Liu, Audris Huang, John Tokarski, Aberra Fura, Thomas Spires, Joh…
Bioorganic & Medicinal Chemistry Letters
Several Non-salt and Solid Thienopyridine Derivatives as Oral P2Y<sub>12</sub> Receptor Inhibitors with Good Stability
Publication date: Available online 1 September 2022Source: Bioorganic & Medicinal Chemistry LettersAuthor(s): Lei Liu, Lingjun Li, Jing Yuan, Wei Liu, Yuquan Li, Shijun Zhang, Changjiang Huang