Bioorganic & Medicinal Chemistry Letters
Graphical Abstract Contents Continued
Publication date: 1 January 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 79Author(s):
Bioorganic & Medicinal Chemistry Letters
Design, synthesis, and bioactivity evaluation of novel 1-(4-(benzylsulfonyl)-2-nitrophenyl) derivatives as potential anti-inflammatory agents against LPS-induced acute lung injury
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 80Author(s): Pan Chen, Yiming Yu, Sijia Su, Zhiteng Du, Binhao Cai, Xiaoyu Sun, Nipon Chattipakorn, Aleksandr V. Samorodov, Valentin N. Pavlov, Qidong Tang, Won-J…
Bioorganic & Medicinal Chemistry Letters
New class of fused [3,2-b][1,2,4]triazolothiazoles for targeting glioma <em>in vitro</em>
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 80Author(s): Papisetti Venkatesham, Nikhil Ranjan, Anwita Mudiraj, Vinutha Kuchana, Raju Chedupaka, Vijjulatha Manga, Phanithi Prakash Babu, Rajeswar Rao Vedula
Bioorganic & Medicinal Chemistry Letters
Synthesis and biological evaluation of <em>N</em>-(benzene sulfonyl)acetamide derivatives as anti-inflammatory and analgesic agents with COX-2/5-LOX/TRPV1 multifunctional inhibitory activity
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 80Author(s): Wenli Chen, Qinlong Xu, Xiaodong Ma, Jiajia Mo, Gaofeng Lin, Guangwei He, Zhaoxing Chu, Jiaming Li
Bioorganic & Medicinal Chemistry Letters
Design, synthesis and biological evaluation of novel 3,4-dihydro-2<em>H</em>-[1,4]oxazino [2,3-<em>f</em>]quinazolin derivatives as EGFR-TKIs
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 80Author(s): Xuemei Qin, Peng Liu, Yihai Li, Liming Hu, Yexin Liao, Tingting Cao, Lifang Yang
Bioorganic & Medicinal Chemistry Letters
Synthesis, anticancer evaluation, and molecular docking studies of thiazolyl-pyrazoline derivatives
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 80Author(s): Narges Hosseini Nasab, Fereshteh Azimian, Rok Su Shim, Young Seok Eom, Fahad Hassan Shah, Song Ja Kim
Bioorganic & Medicinal Chemistry Letters
Persistent challenges in the development of an mGlu<sub>7</sub> PAM <em>in vivo</em> tool compound: The discovery of VU6046980
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 80Author(s): Jacob J. Kalbfleisch, Alice L. Rodriguez, Xia Lei, Kelly Weiss, Annie L. Blobaum, Olivier Boutaud, Colleen M. Niswender, Craig W. Lindsley
Bioorganic & Medicinal Chemistry Letters
Synthesis and biological activity evaluation of novel 3,5,7-trisubstituted pyrazolo[1,5-<em>a</em>]pyrimidines
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 80Author(s): Kristýna Vlková, Růžena Padrtová, Tomáš Gucký, Miroslav Peřina, Eva Řezníčková, Vladimír Kryštof
Bioorganic & Medicinal Chemistry Letters
A concise review on marine bromopyrrole alkaloids as anticancer agents
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 80Author(s): Safia Mahamed, Raeesa Motal, Titus Govender, Nompilo Dlamini, Kwanele Khuboni, Zamahlubi Hadeb, Baji Baba Shaik, Kimeshni Moodley, Sachin Balaso Mohi…
Bioorganic & Medicinal Chemistry Letters
Novel imidazo[1,5-<em>a</em>]quinoxaline derivatives: SAR, selectivity and modeling challenges en route to the identification of an α5-GABAA receptor NAM
Publication date: 15 January 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 80Author(s): Benedek Imre Károlyi, Attila Potor, Gábor László Kapus, László Fodor, Amrita Bobok, Balázs Krámos, Ildikó Magdó, Imre Bata, György Szabó