Bioorganic & Medicinal Chemistry Letters
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Publication date: 15 July 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 91Author(s):
Bioorganic & Medicinal Chemistry Letters
Design, synthesis and evaluation of new pyrimidine derivatives as EGFR<sup>C797S</sup> tyrosine kinase inhibitors
Publication date: 15 July 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 91Author(s): Yu-Ze Mao, Xiao-Xiao Xi, Hong-Yi Zhao, Yin-Liang Zhang, San-Qi Zhang
Bioorganic & Medicinal Chemistry Letters
Graphical Abstract TOC
Publication date: 15 July 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 91Author(s):
Bioorganic & Medicinal Chemistry Letters
Design and synthesis of aminopyridine containing biaryls reducing c-MYC protein levels in cells
Publication date: 15 August 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 92Author(s): Christina N. Di Marco, Lamont Terrell, Robert Sanchez, Lourdes Rueda, Leanna Shuster, Eldridge N. Nartey, Charles McHugh, James F. Mack, Arthur Shu, X…
Bioorganic & Medicinal Chemistry Letters
Synthesis of proposed structure of ledebourin A
Publication date: 15 August 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 92Author(s): Seunggyu Jeon, Seul Lee, Minkyu Ji, Md. Samsuzzaman, Sangil Kwon, Sun Yeou Kim, Seung-Yong Seo
Bioorganic & Medicinal Chemistry Letters
Discovery of potent NAMPT-Targeting PROTACs using FK866 as the warhead
Publication date: 15 August 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 92Author(s): Peifeng Zhang, Wei Wang, Menglu Guo, Luozhu Zhou, Guoqiang Dong, Defeng Xu, Chunquan Sheng
Bioorganic & Medicinal Chemistry Letters
Synthesis, activity, metabolic stability and cell permeability of new cytosolic phospholipase A<sub>2</sub>α inhibitors with 1-indolyl-3-phenoxypropan-2-one structure
Publication date: 15 August 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 92Author(s): Angelina Subeska, Merlin Ekodo Voundi, Walburga Hanekamp, Dennis Mulac, Klaus Langer, Matthias Lehr
Bioorganic & Medicinal Chemistry Letters
In vivo variable and multi-day response from an insulin-releasing photoactivated depot
Publication date: 15 August 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 92Author(s): Karthik Nadendla, Swetha Chintala, Karen Kover, Simon H. Friedman
Bioorganic & Medicinal Chemistry Letters
Discovery of 5-((1H-indazol-3-yl) methylene)-2-thioxoimidazolidin-4-one derivatives as a new class of AHR agonists with anti-psoriasis activity in a mouse model
Publication date: 15 August 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 92Author(s): Guo Zhang, Ziyi Xia, Chenyu Tian, Anjie Xia, Jing You, Jie Liu, Shengyong Yang, Linli Li
Bioorganic & Medicinal Chemistry Letters
Design, synthesis and biological evaluation of nitric oxide-releasing 5-cyano-6-phenyl-2, 4-disubstituted pyrimidine derivatives
Publication date: 15 August 2023Source: Bioorganic & Medicinal Chemistry Letters, Volume 92Author(s): Lingling Chi, Hao Wang, Fuqiang Yu, Chao Gao, Honglin Dai, Xiaojie Si, Yuze Dong, Hongmin Liu, Qiurong Zhang