September 2023

Synthesis of 1,3,5-triphenyl-1,2,4-triazole derivatives and their neuroprotection by anti-oxidative stress and anti-inflammation and protecting BBB

Publication date: 15 November 2023Source: European Journal of Medicinal Chemistry, Volume 260Author(s): Yang Wang, Ruiqi Su, Jianwen Chen, Xuan Liu, Jingning Luo, Yaoqiang Lao, Ping Huang, Jinguo Shi, Caibao Jiang, Liping Liao, Jingxia Zhang

By ScienceDirect Publication: European Journal of Medicinal Chemistry, ago

Synthesis and evaluation of 2-NMPA derivatives as potential agents for prevention of osteoporosis <em>in vitro</em> and <em>in vivo</em>

Publication date: 15 November 2023Source: European Journal of Medicinal Chemistry, Volume 260Author(s): Zhihao Chen, Devaneyan Joseph, Mina Ding, Swapnil Pandurang Bhujbal, Robin Prakash Sirvin Rajan, Eunae Kim, Sang-wook Park, Sunwoo Lee, Tae-Hoon Lee

By ScienceDirect Publication: European Journal of Medicinal Chemistry, ago

Cantharidin analogue alleviates dextran sulfate sodium-induced colitis in mice by inhibiting the activation of NF-κB signaling

Publication date: 15 November 2023Source: European Journal of Medicinal Chemistry, Volume 260Author(s): Yihang Wu, Zixiu Liu, Zhenxiu He, Jumei Yi, Xingfang Qiao, Chunbin Tan, Yajing Xing, Yaobo Zeng, Dajian Yang, Junlin Yin, Baomin Fan, Guangzhi Zeng

By ScienceDirect Publication: European Journal of Medicinal Chemistry, ago

Lead generation from <em>N</em>-[benzyl(4-phenylbutyl)carbamoyl]amino acid as a novel LPA<sub>1</sub> antagonist for the treatment of systemic sclerosis

Publication date: 15 November 2023Source: European Journal of Medicinal Chemistry, Volume 260Author(s): Yuki Kobayashi, Fumito Uneuchi, Takumi Naruse, Daisuke Matsuda, Lisa Okumura-Kitajima, Hiromitsu Kajiyama, Reiko Wada, Yuki Yonemoto, Koichiro Nakan…

By ScienceDirect Publication: European Journal of Medicinal Chemistry, ago

Novel spiro[pyrrolidine-2,3′-quinoline]-2′-one derivatives containing piperazine fragment as potential chitin synthase inhibitors and antifungal agents: Design, synthesis and biological evaluation

Publication date: 15 November 2023Source: European Journal of Medicinal Chemistry, Volume 260Author(s): Lige Liu, Hu Wu, Yan Long, Xinlong Yang, Chuanbiao Du, Yajie Xu, Qinggang Ji

By ScienceDirect Publication: European Journal of Medicinal Chemistry, ago