March 2023

3,4-Dihydrobenzo[e][1,2,3]oxathiazine 2,2-dioxide analogs act as potential AMPA receptor potentiators with antidepressant activity

Publication date: 5 May 2023Source: European Journal of Medicinal Chemistry, Volume 251Author(s): Long wei, Xueyu Qi, Xueli Yu, Yanghao Zheng, Xing Luo, Yingying Wei, Peiyan Ni, Liansheng Zhao, Qiang Wang, Xiaohong Ma, Wei Deng, Wanjun Guo, Xun Hu, Tao Li

By ScienceDirect Publication: European Journal of Medicinal Chemistry, ago

Discovery of a novel 1<em>H</em>-pyrazole- [3,4-b] pyridine-based lysine demethylase 5B inhibitor with potential anti-prostate cancer activity that perturbs the phosphoinositide 3-kinase/AKT pathway

Publication date: 5 May 2023Source: European Journal of Medicinal Chemistry, Volume 251Author(s): Yaquan Cao, Pu Yang, Yingxue Yang, Zihui Lin, Zhengmin Fan, Xuliang Wei, Lijie Yan, Yongchun Li, Zhangxu He, Liying Ma, Hongde Xu, Chunli Wu

By ScienceDirect Publication: European Journal of Medicinal Chemistry, ago

Design, synthesis, and repurposing of <em>O</em><sup><em>6</em></sup>-aminoalkyl-sulfuretin analogs towards discovery of potential lead compounds as antileishmanial agents

Publication date: 5 May 2023Source: European Journal of Medicinal Chemistry, Volume 251Author(s): Ahmed H.E. Hassan, Trong-Nhat Phan, Suyeon Moon, Chae Hyeon Lee, Yeon Ju Kim, Soo Bin Cho, Selwan M. El-Sayed, Yeonwoo Choi, Joo Hwan No, Yong Sup Lee

By ScienceDirect Publication: European Journal of Medicinal Chemistry, ago